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- Publisher
- Springer Journals
- Copyright
- Copyright © 2015 by Springer Science+Business Media Dordrecht
- Subject
- Chemistry; Catalysis; Physical Chemistry; Inorganic Chemistry
- ISSN
- 0922-6168
- eISSN
- 1568-5675
- DOI
- 10.1007/s11164-014-1835-y
- Publisher site
- See Article on Publisher Site
Abstract
A series of novel neonicotinoids containing a dihydro-pyridine ring and a trifluoromethyl group were designed and synthesized by multicomponent reactions of 6-Cl-PMNI, triethoxymethane and 4,4,4-trifluoro-3-oxobutaneanilides (9) under solvent-free and catalyst-free conditions. The trifluoromethyl group plays an important role as an electron-withdrawing group in enhancing the reaction activity of compound 9. The target compounds were characterized by 1H NMR, IR and elemental analysis. Bioassays indicated that most of the synthesized compounds exhibited moderate insecticidal activities against Aphis craccivora.
Journal
Research on Chemical Intermediates – Springer Journals
Published: Feb 17, 2015