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in considering its antiparkinsonian effects, or an exclusive role of 5 - HT 2A/ 2C receptor activation in hallucinogenesis. These conclusions are surprising when one considers that the potent interaction of lisuride ...
. Brexpiprazole is a novel serotonin-dopamine activity modulator that acts as a partial agonist of serotonin 1A ( 5 -HT1A) and dopamine D2 receptors , as well as a potent antagonist of 5 -HT2A receptors ...
These results indicate that aripiprazole modulates the in vivo 5 - HT and DA release in mPFC through the activation of 5 - HT 1A receptors . Moreover, aripiprazole behaves as a partial agonist at DA D2 ...
), a selective 5 -HT1A receptor agonist , and 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane (DOI), a selective 5 -HT2A/ 2C receptor agonist , on the performance of middle-aged rats in a two-lever choice reaction task ...
patient. Brexpiprazole is a serotonin–dopamine activity Otsuka Pharmaceutical Co., Ltd., Tokyo, modulator: a partial agonist at 5 - HT and dopamine D receptors at similar potency, Japan 1A 2 4 ...
1 depression (June 2013). Lurasidone has a strong antagonistic property at the D2, serotonin ( 5 - HT )2A, and 5 -HT7 receptors , and partial agonistic property at the 5 -HT1A receptor . Lurasidone also has ...
was an antagonist at 5 -HT2A, 5 -HT2B, 5 -HT2C, α 1A , α 1D, α 2A, α 2C , H1, M1, M3, and M5 receptors . In the mouse tail suspension test, N-Desalkylquetiapine displayed potent antidepressant-like activity in VMAT2 ...
-HT2B-, hD2L-, and hD3-dopamine receptors , but also has significant affinity ( 5 –30 nM) for several other 5 - HT receptors ( 5 -HT1A, 5 -HT2A, 5 -HT7), as well as α 1A -adrenergic and hH1-histamine receptors ...
2A ( 5 ‐ HT 2A ), 5 ‐ HT 1A , 5 ‐ HT 7 , and noradrenaline alpha‐ 2C (α 2c ) receptors , displaying antagonist activity at 5 ‐ HT 7 receptors and moderate partial agonist activity at 5 ‐ HT 1A receptors (Ishibashi ...
of these receptors in the response. In contrast, the 5 -HTR4 agonist cisapride significantly increased PRL secretion. The 5 - HT agonist , α-methyl- 5 - HT , which preferentially activates the 5 -HTR2 subtypes (48, 53, 54, 67 ...
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