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Pharmacological activities of some triazinopyrazolothieno pyrimidine derivatives

Pharmacological activities of some triazinopyrazolothieno pyrimidine derivatives REFERENCES1. A. B. Siddiqui, A. R. Trivedi, V. B. Kataria and V. H. Shah, 4,5-Dihydro-1H-pyrazolo[3,4-d]pyrimidine containing phenothiazines as antitubercular agents, Bioorg. Med. Chem. Lett. 51 (2014) 1493–1495; DOI: 10.1016/j.bmcl.2014.02.012.10.1016/j.bmcl.2014.02.0122. N. M. Y. Elsayed, D. A. Abou El Ella, R. A. T. Serya, M. F. Tolba, R. Shalaby and K. A. M. Abouzid, Design, synthesis and biological evaluation of indazole-pyrimidine based derivatives as anticancer agents with anti-angiogenic and antiproliferative activities, Med. Chem. Commun. 7 (2016) 881–899; DOI: 10.1039/C5MD00602C.10.1039/C5MD00602C3. A. K. Verma, R. Kumari, A. K. Sing, B. B. Sharma, A. Martin and R. Kant, Synthesis characterization and anticancer activity of novel N-(sugar pyranosyl)thienopyrimidine 4-amine derivatives, Int. Res. J. Pharm. 5 (2014) 922–925; DOI: 10.7897/2230-8407.0512187.10.7897/2230-8407.05121874. S. Kumaresan, S. Chandrasekaran, K. M. Sakthivel, C. Guruvayoorappan and V. M. Israel, Synthesis, characterization and anti-inflammatory activity of some novel pyrimidin-2-amines on carrageenan-induced paw edema in balb/c mice, J. Chem. Pharm. Res. 6 (2014) 593–606.5. H. J. Zhang, S. B. Wang, X. Wen, J. Z. Li and Z. S. Quan, Design, synthesis, and evaluation of the anticonvulsant and antidepressant activities of pyrido[2,3-d]pyrimidine derivatives, Med. Chem. Res. 25 (2016) 1287–1298; DOI: 10.1007/s00044-016-1559-1.http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000378573400001&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f310.1007/s00044-016-1559-16. K. Singh, H. Kaur, K. Chibale, J. Balzarini, S. Little and P. V. Bharatam, 2-Aminopyrimidine based 4-aminoquinoline anti-plasmodial agents. Synthesis, biological activity, structure-activity relationship and mode of action studies, Eur. J. Med. Chem. 52 (2012) 82–97; DOI: 10.1016/j.ejmech.2012.03.007.10.1016/j.ejmech.2012.03.007http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000304291600009&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f37. A. A. Abu-Hashem and M. M. Youssef, Synthesis of new visnagen and khellin furochromone pyrimidine derivatives and their anti-inflammatory and analgesic activity, Molecules 16 (2011) 1956–1972; DOI: 10.3390/molecules16031956.10.3390/molecules16031956http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000288853400003&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f38. P. Rathee, R. K. Tonk, A. Dalal, M. K. Ruhil and A. Kumar, Synthesis and application of thiobarbituric acid derivatives as antifungal agents, Cell. Mol. Biol. 62 (2016) 5 pages; DOI: 10.4172/1165-158X.1000141.10.4172/1165-158X.10001419. D. Cai, Z.-H. Zhang, Y. Chen, X.-J. Yan, S.-T. Zhang, L.-J. Zou, L.-H. Meng, F. Li and B.-J. Fu, Synthesis of some new thiazolo[3,2-a]pyrimidine derivatives and screening of their in vitro antibacterial and antitubercular activities, Med. Chem. Res. 25 (2016) 292–302; DOI: 10.1007/s00044-015-1481-y.http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000368548800008&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f310.1007/s00044-015-1481-y10. N. O. Al-Harbi, S. A. Bahashwan, A. A. Fayed, M. S. Aboonq, A. El-Galil and E. Amr, Anti-parkinsonism, hypoglycemic and anti-microbial activities of new poly fused ring heterocyclic candidates, Int. J. Biol. Macromol. 57 (2013) 165–173; DOI: 10.1016/j.ijbiomac.2013.03.019.http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000319098900026&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f310.1016/j.ijbiomac.2013.03.01911. S. A. Bahashwan, N. O. Al-Harbi, A. Fayed, A. El-Galil E. Amr, K. Shadid, A. M. Alalawi and I. M. S. Bassati, Pharmacological activities of some new polycyclic triazolopyrazolopyridazine derivatives, Int. J. Biol. Macromol. 51 (2012) 7–17; DOI: 10.1016/j.ijbiomac.2012.05.002.http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000306038600002&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f310.1016/j.ijbiomac.2012.05.00212. S. A. Bahashwan, A. A. Fayed, A. El-Galil E. Amr, E. M. Flefel and A. Kalmouch, Synthesis and pharmacological activities of some new triazolo- and tetrazolopyrimidine derivatives, Molecules 18 (2013) 15051–15063; DOI: 10.3390/molecules181215051.10.3390/molecules181215051http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000330315700039&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f313. A. N. O. Al-Harbi, S. A. Bahashwan, A. A. Fayed and M. A. Ramadan, Pharmacological activities evaluation of some new pyrazolo-pyrimidino-pyridazine derivatives, Afr. J. Pharm. Pharmacol. 7 (2013) 517–523; DOI: 10.5897/AJPPX12.003.10.5897/AJPPX12.00314. A. L. A. Lima, A. F. Alves, A. L. Xavier, T. Mozzini-Monteiro, T. R. R. Oliveira, F. C. Leite, M. H. Shih and F. Y. Ke, Syntheses and evaluation of antioxidant activity of sydnonyl substituted thiazolidinone and thiazoline derivatives, Bioorg. Med. Chem. 12 (2004) 4633–4643; DOI: 10.1016/j.bmc.2004.06.033.10.1016/j.bmc.2004.06.03315. W. N. Matias, M. M. V. S. C. Branco, M. F. V. Souza and M. R. Piuvezam, Anti-inflammatory activity and acute toxicity studies of hydroalcoholic extract of Herissantia tiubae, Bras. J. Pharmacogn. 26 (2016) 225–232; DOI: 10.1016/j.bjp.2015.11.001.10.1016/j.bjp.2015.11.001 http://www.deepdyve.com/assets/images/DeepDyve-Logo-lg.png Acta Pharmaceutica de Gruyter

Pharmacological activities of some triazinopyrazolothieno pyrimidine derivatives

Bahashwan, Saleh A.
Acta Pharmaceutica , Volume 67 (3): 8 – Sep 1, 2017
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Publisher
de Gruyter
Copyright
© 2017 Saleh A. Bahashwan, published by De Gruyter Open
ISSN
1846-9558
eISSN
1846-9558
DOI
10.1515/acph-2017-0022
pmid
28858840
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Abstract

REFERENCES1. A. B. Siddiqui, A. R. Trivedi, V. B. Kataria and V. H. Shah, 4,5-Dihydro-1H-pyrazolo[3,4-d]pyrimidine containing phenothiazines as antitubercular agents, Bioorg. Med. Chem. Lett. 51 (2014) 1493–1495; DOI: 10.1016/j.bmcl.2014.02.012.10.1016/j.bmcl.2014.02.0122. N. M. Y. Elsayed, D. A. Abou El Ella, R. A. T. Serya, M. F. Tolba, R. Shalaby and K. A. M. Abouzid, Design, synthesis and biological evaluation of indazole-pyrimidine based derivatives as anticancer agents with anti-angiogenic and antiproliferative activities, Med. Chem. Commun. 7 (2016) 881–899; DOI: 10.1039/C5MD00602C.10.1039/C5MD00602C3. A. K. Verma, R. Kumari, A. K. Sing, B. B. Sharma, A. Martin and R. Kant, Synthesis characterization and anticancer activity of novel N-(sugar pyranosyl)thienopyrimidine 4-amine derivatives, Int. Res. J. Pharm. 5 (2014) 922–925; DOI: 10.7897/2230-8407.0512187.10.7897/2230-8407.05121874. S. Kumaresan, S. Chandrasekaran, K. M. Sakthivel, C. Guruvayoorappan and V. M. Israel, Synthesis, characterization and anti-inflammatory activity of some novel pyrimidin-2-amines on carrageenan-induced paw edema in balb/c mice, J. Chem. Pharm. Res. 6 (2014) 593–606.5. H. J. Zhang, S. B. Wang, X. Wen, J. Z. Li and Z. S. Quan, Design, synthesis, and evaluation of the anticonvulsant and antidepressant activities of pyrido[2,3-d]pyrimidine derivatives, Med. Chem. Res. 25 (2016) 1287–1298; DOI: 10.1007/s00044-016-1559-1.http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000378573400001&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f310.1007/s00044-016-1559-16. K. Singh, H. Kaur, K. Chibale, J. Balzarini, S. Little and P. V. Bharatam, 2-Aminopyrimidine based 4-aminoquinoline anti-plasmodial agents. Synthesis, biological activity, structure-activity relationship and mode of action studies, Eur. J. Med. Chem. 52 (2012) 82–97; DOI: 10.1016/j.ejmech.2012.03.007.10.1016/j.ejmech.2012.03.007http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000304291600009&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f37. A. A. Abu-Hashem and M. M. Youssef, Synthesis of new visnagen and khellin furochromone pyrimidine derivatives and their anti-inflammatory and analgesic activity, Molecules 16 (2011) 1956–1972; DOI: 10.3390/molecules16031956.10.3390/molecules16031956http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000288853400003&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f38. P. Rathee, R. K. Tonk, A. Dalal, M. K. Ruhil and A. Kumar, Synthesis and application of thiobarbituric acid derivatives as antifungal agents, Cell. Mol. Biol. 62 (2016) 5 pages; DOI: 10.4172/1165-158X.1000141.10.4172/1165-158X.10001419. D. Cai, Z.-H. Zhang, Y. Chen, X.-J. Yan, S.-T. Zhang, L.-J. Zou, L.-H. Meng, F. Li and B.-J. Fu, Synthesis of some new thiazolo[3,2-a]pyrimidine derivatives and screening of their in vitro antibacterial and antitubercular activities, Med. Chem. Res. 25 (2016) 292–302; DOI: 10.1007/s00044-015-1481-y.http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000368548800008&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f310.1007/s00044-015-1481-y10. N. O. Al-Harbi, S. A. Bahashwan, A. A. Fayed, M. S. Aboonq, A. El-Galil and E. Amr, Anti-parkinsonism, hypoglycemic and anti-microbial activities of new poly fused ring heterocyclic candidates, Int. J. Biol. Macromol. 57 (2013) 165–173; DOI: 10.1016/j.ijbiomac.2013.03.019.http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000319098900026&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f310.1016/j.ijbiomac.2013.03.01911. S. A. Bahashwan, N. O. Al-Harbi, A. Fayed, A. El-Galil E. Amr, K. Shadid, A. M. Alalawi and I. M. S. Bassati, Pharmacological activities of some new polycyclic triazolopyrazolopyridazine derivatives, Int. J. Biol. Macromol. 51 (2012) 7–17; DOI: 10.1016/j.ijbiomac.2012.05.002.http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000306038600002&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f310.1016/j.ijbiomac.2012.05.00212. S. A. Bahashwan, A. A. Fayed, A. El-Galil E. Amr, E. M. Flefel and A. Kalmouch, Synthesis and pharmacological activities of some new triazolo- and tetrazolopyrimidine derivatives, Molecules 18 (2013) 15051–15063; DOI: 10.3390/molecules181215051.10.3390/molecules181215051http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcApp=PARTNER_APP&SrcAuth=LinksAMR&KeyUT=WOS:000330315700039&DestLinkType=FullRecord&DestApp=ALL_WOS&UsrCustomerID=b7bc2757938ac7a7a821505f8243d9f313. A. N. O. Al-Harbi, S. A. Bahashwan, A. A. Fayed and M. A. Ramadan, Pharmacological activities evaluation of some new pyrazolo-pyrimidino-pyridazine derivatives, Afr. J. Pharm. Pharmacol. 7 (2013) 517–523; DOI: 10.5897/AJPPX12.003.10.5897/AJPPX12.00314. A. L. A. Lima, A. F. Alves, A. L. Xavier, T. Mozzini-Monteiro, T. R. R. Oliveira, F. C. Leite, M. H. Shih and F. Y. Ke, Syntheses and evaluation of antioxidant activity of sydnonyl substituted thiazolidinone and thiazoline derivatives, Bioorg. Med. Chem. 12 (2004) 4633–4643; DOI: 10.1016/j.bmc.2004.06.033.10.1016/j.bmc.2004.06.03315. W. N. Matias, M. M. V. S. C. Branco, M. F. V. Souza and M. R. Piuvezam, Anti-inflammatory activity and acute toxicity studies of hydroalcoholic extract of Herissantia tiubae, Bras. J. Pharmacogn. 26 (2016) 225–232; DOI: 10.1016/j.bjp.2015.11.001.10.1016/j.bjp.2015.11.001

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Acta Pharmaceutica – de Gruyter

Published: Sep 1, 2017

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