TY - JOUR
AU1 - RICOUART, ANNIE
AU2 - MAES, PIERRETTE
AU3 - BATTMANN, THIERRY
AU4 - KERDELHUE, BERNARD
AU5 - TARTAR, ANDRÉ
AU6 - SERGHERAERT, CHRISTIAN
AB - Beyond its aromatic character and important hydrophobicity, cymantrenylalanine, a metallocenic amino‐acid, can be easily photosubstituted with phosphine and phosphite ligands to readily yield new analogs with different hydrophobicity and steric hindrance. The incorporation of phosphine and phosphite ligands is described. As an illustration of the offered possibilities, the synthesis and the biological activity of two new GnRH analogs modified in position 6 are reported.
TI - Photosubstitution of cymantrenylalanine as a tool in peptide chemistry
JF - Chemical Biology & Drug Design
DO - 10.1111/j.1399-3011.1988.tb00926.x
DA - 1988-07-01
UR - https://www.deepdyve.com/lp/wiley/photosubstitution-of-cymantrenylalanine-as-a-tool-in-peptide-chemistry-27TiToP8YX
SP - 56
EP - 63
VL - 32
IS - 1
DP - DeepDyve
ER -